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Updated: Aug 17, 2026

A Fluorescent Screening Assay for Identifying Modulators of GIRK Channels
05:31

A Fluorescent Screening Assay for Identifying Modulators of GIRK Channels

Published on: April 24, 2012

組合せ化学によるソマトスタチン受容体の亜型選択性アゴニストの迅速な特定

S P Rohrer1, E T Birzin, R T Mosley

  • 1Department of Cell Biochemistry and Physiology, Merck Research Laboratories, Post Office Box 2000, Rahway, NJ 07065, USA. susanvrohrer@merck.com

Science (New York, N.Y.)
|October 23, 1998
PubMed
まとめ

研究者らはソマトスタチン受容体の非ペプチドアゴニストを開発し,グルカゴン,インスリン,成長ホルモン放出を調節するソマトスタチンサブタイプ-2および-5受容体の役割を明らかにした.

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