Cheminformatics and quantitative structure-activity relationships
Recently Published Articles
Gallic Acid-Rich Ephedra alata: Integrated Phytochemical Profiling, Aromatase Docking, and Optimized Extraction via Box-Behnken Design
Nadjat Chekroun-Bechlaghem, Nabila Belyagoubi-Benhammou, Zineb Kaid, Amel Zitouni, Imad Abdelhamid El Haci, Abdelghani Bouchama, Ahmed Djafri
Development and Characterization of a Topical Spray Containing <i>Channa striata</i> and <i>Anredera cordifolia</i> Extracts for Wound Healing: <i>In Vivo</i> Evaluation in Mices
Heru Sasongko, M H N Putro
Design, Synthesis, and Structure-Activity Relationship Studies of Novel 3CL<sup>pro</sup> Inhibitors
Yixuan Feng, Feng Wang, Donglan Liu, Qiqi Yan, Leyuan Kang, Wenhao Zhao, Shixin Jin, Shuxiang Huang, Jincun Zhao, Ping Tian, Dingding Gao
Potential c-Met-targeted pyrazole-pyridine-oxadiazole hybrids: synthesis, anticancer activity, and computational rationale
Prince A Dave, Jay B Maheta, Darshna K Lakhnotra, Nargis H Shaikh, Ila M Ram, Chintan P Somaiya, Tarun Parangi, Yogesh O Bhola
Study on Synthesis, Antiproliferative Properties, Immunomodulatory Effects, and Anti-Breast Cancer Activity of New Δ<sup>2</sup>-Pyrazoline-1H-1,2,3-Triazole Derivatives
Sadiq Noor Khan, Hassan Moghtaderi, Ebrahimi Amirhossein, Saeed Mohammadi, Satya Kumar Avula, Sobia Ahsan Halim, Shahid Duran, Najeeb Ur Rehman, Shaikh Mizanoor Rahman, Ajmal Khan, René Csuk, Ali Rostami, Ahmed Al-Harrasi
Discovery of Virulence Attenuator of Chromobacterium violaceum CV026 From Marine-Derived Fungus Aspergillus ochraceus LSD-13 by Inhibiting Quorum Sensing and Destroying Biofilm
Xinyi Li, Hui Wang, Yibo Wu, Xiaohan Ding, Shurong Guo, Shuang Gao, Shiwei Sun, Wei Wang
Discovery of 4-aminochalcone-based dual α-glucosidase and aldose reductase inhibitors: <i>in vitro</i>, <i>in vivo</i>, and <i>in silico</i> studies
Ehsan Ullah Mughal, Nafeesa Naeem, Songül Bayrak, Namık Kılınç, Bushra Shakoor, Magdi E A Zaki, Maher Fathalla, Sobhi M Gomha, Amina Sadiq, Züleyha Almaz
Identification and structure-activity relationship studies of clavatol as an antifungal compound against pathogenic plant fungi using a drug-hypersensitive fission yeast screening system
Aoi Kimishima, Sota Negami, Wakana Yoda, Taichi Kamo, Sota Honma, Shigehiro A Kawashima, Yoko Yashiroda, Paul Wasuwanich, Yukiko Ujie, Shin-Ichi Fuji, Toshiyuki Tokiwa, Hiroki Kojima, Akihiro Sugawara, Takumi Chinen, Takeo Usui, Yukihiro Asami