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对选择性甲状腺激素受体调节器的哈梅特分析揭示了对激素抗剂的结构和电子要求

Ngoc-Ha Nguyen1, James W Apriletti, John D Baxter

  • 1Program in Chemistry and Chemical Biology, Department of Pharmaceutical Chemistry, University of California-San Francisco, San Francisco, CA 94143-0446, USA.

Journal of the American Chemical Society
|March 31, 2005
PubMed
概括

选择性甲状腺激素受体 (TR) 调节剂具有治疗潜力. 研究人员发现,特定的电子性质,不一定是基,是新型化合物中TR抗体活性的关键.

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