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Updated: Jul 4, 2026

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单甲基素与Zn2+在葡萄糖皮质类受体的结合部位上竞争

Anne M Spuches1, Dean E Wilcox

  • 1Department of Chemistry, Dartmouth College, Hanover, New Hampshire 03755, USA.

Journal of the American Chemical Society
|June 6, 2008
PubMed
概括

单甲基化 (MMAIII),与化不同,将离子从葡萄糖皮质体受体DNA结合域 (GR-DBD) 中取代. 这种干扰会损害受体结合DNA的能力,影响基因调节.

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