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Updated: Jun 23, 2026

Methods for Evaluating the Role of c-Fos and Dusp1 in Oncogene Dependence
10:09

Methods for Evaluating the Role of c-Fos and Dusp1 in Oncogene Dependence

Published on: January 7, 2019

小分子抑制剂在蛋白c-Myc上存在多个独立的结合点

Dalia I Hammoudeh1, Ariele Viacava Follis, Edward V Prochownik

  • 1Department of Chemistry, Georgetown University, Washington, District of Columbia 20057, USA.

Journal of the American Chemical Society
|May 13, 2009
PubMed
概括

研究人员确定了小分子抑制剂的c-Myccoprotein上三个不同的结合点. 这些位点允许同时独立结合,保存c-Myc.

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Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors10:33

Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors

Published on: October 26, 2015

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