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Updated: Jun 16, 2026

Preparation of Stable Bicyclic Aziridinium Ions and Their Ring-Opening for the Synthesis of Azaheterocycles
11:45

Preparation of Stable Bicyclic Aziridinium Ions and Their Ring-Opening for the Synthesis of Azaheterocycles

Published on: August 22, 2018

角替代的1-azabicyclic环系统的选合成:使用aza-Cope重排的动态动态分辨率

Tatsuya Ito1, Larry E Overman, Jocelyn Wang

  • 1Department of Chemistry, University of California, Irvine, 1102 Natural Sciences II, Irvine, California 92697-2025, USA.

Journal of the American Chemical Society
|February 24, 2010
PubMed
概括

一种新型的酶选择性合成提供了角度替代的1-azabicyclic amines,具有高产率和99%的酶因子过量 (ee). 这种方法利用独特的动态动力学分辨率策略来实现高效的立体选择合成.

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