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Updated: Jun 3, 2026

Preparation of Stable Bicyclic Aziridinium Ions and Their Ring-Opening for the Synthesis of Azaheterocycles
11:45

Preparation of Stable Bicyclic Aziridinium Ions and Their Ring-Opening for the Synthesis of Azaheterocycles

Published on: August 22, 2018

替代型皮佩里丁的高度二元选择性亚里लेशन

Stephanie Seel1, Tobias Thaler, Keishi Takatsu

  • 1Department Chemie, Ludwig-Maximilians-Universität München, Butenandtstr. 5-13, Haus F, 81377 Munich, Germany.

Journal of the American Chemical Society
|March 11, 2011
PubMed
概括

一种新的方法使用Negishi交叉合来创建具有高立体选择性的替代皮佩里丁. 这种方法控制了 cis 或 trans 异构体的形成,从而精确控制了 piperidine 的合成.

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