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激动剂结合的神经酶受体的结构

Jim F White1, Nicholas Noinaj, Yoko Shibata

  • 1Membrane Protein Structure Function Unit, National Institute of Neurological Disorders and Stroke, National Institutes of Health, Department of Health and Human Services, Rockville, Maryland 20852, USA.

Nature
|October 12, 2012
PubMed
概括

研究人员确定了与其激活器结合的神经素受体1 (NTSR1) 的结构. 这为-GPCR结合提供了第一个洞察力,有助于开发用于神经系统疾病,癌症和肥胖症的药物.

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