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Updated: May 16, 2026

Preparation and In Vivo Use of an Activity-based Probe for N-acylethanolamine Acid Amidase
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Preparation and In Vivo Use of an Activity-based Probe for N-acylethanolamine Acid Amidase

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在脂肪酸胺基酸酶中,非类固醇抗炎药物的结合部位

Laura Bertolacci1, Elisa Romeo, Marina Veronesi

  • 1Drug Discovery and Development, Istituto Italiano di Tecnologia, Via Morego 30, 16163 Genoa, Italy.

Journal of the American Chemical Society
|December 18, 2012
PubMed
概括

非类固醇抗炎药物 (NSAIDs) 可以阻断脂肪酸胺酸酶 (FAAH),这是一种降解内分泌素的酶. 这种双重作用可能会通过结合NSAID和内分泌大麻素路径效应来改善疼痛缓解.

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