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Updated: Jan 19, 2026

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混合炸弹在类似物中:在定义的距离内结合激动剂和对抗剂,以优化瘤向

Carsten Kroll1, Rosalba Mansi, Friederike Braun

  • 1Laboratory of Organic Chemistry, ETH Zürich , Zürich, Switzerland.

Journal of the American Chemical Society
|November 2, 2013
PubMed
概括

研究人员开发了针对胃素释放受体的新型放射性标记混合配体,以改善瘤成像. 结合体元素之间的20 Å距离显示出较高的前列腺癌细胞吸收和保留.

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