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Updated: Mar 7, 2026

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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替代的2-氨基胺 选择性对α7-尼古丁性乙胆受体激活和与乙胆结合蛋白的关联

Katarzyna Kaczanowska1, Gisela Andrea Camacho Hernandez1,2, Larissa Bendiks1

  • 1Department of Pharmacology, Skaggs School of Pharmacy & Pharmaceutical Sciences, University of California, San Diego , La Jolla, California 92093-0650, United States.

Journal of the American Chemical Society
|February 22, 2017
PubMed
概括

研究人员开发了激活α7尼古丁乙胆受体 (α7-nAChR) 的新型2-氨基胺. 这些化合物具有特定的结合性,为针对尼古丁乙胆受体的新疗法提供了潜力.

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