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Updated: Dec 14, 2025

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甲基转移酶的过渡状态类似物

Niusha Mahmoodi1, Rajesh K Harijan1, Vern L Schramm1

  • 1Department of Biochemistry, Albert Einstein College of Medicine, New York, New York 10461, United States.

Journal of the American Chemical Society
|July 25, 2020
PubMed
概括

甲胺N-甲基转移酶 (PNMT) 抑制剂的设计是为了模仿其过渡状态. 一种新型抑制剂显示纳米分子亲和力,为PNMT相关疾病提供新的治疗潜力.

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