通过Catellani反应进行C-Aryl Glycosides的模块化和立体选择性合成

Weiwei Lv1, Yanhui Chen1, Si Wen1

  • 1College of Materials Science & Engineering, Huaqiao University, Xiamen 361021, China.

概括

这项研究引入了一种新的Catellani型C-H糖化,用于立体选择性地合成多种α-C-基糖化物. 该方法在药物发现中提供了灵活的终止选择和应用,包括达帕格利弗洛辛类似物.

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