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Measuring G-protein-coupled Receptor Signaling via Radio-labeled GTP Binding
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调节G蛋白激活,电流和阿片类受体酸化由pH依赖的抗受体激动剂NFEPP

Melih Özgür Celik1, Viola Seitz1, Fatih Yergöz1

  • 1Department of Experimental Anesthesiology, Charité - Universitätsmedizin Berlin, Corporate Member of Freie Universität Berlin and Humboldt-Universität zu Berlin, Berlin, Germany.

Frontiers in molecular neuroscience
|May 30, 2023
PubMed
概括

通过向酸性组织中的mu-opioid受体 (MOR),N-(3-fluoro-1-phenethylpiperidine-4-yl) -N-phenyl propionamide (NFEPP) 有效地减少疼痛. 这种新型的止痛药可以缓解疼痛.

关键词:
没有NFEPP,没有NFEPP.在VDCC中,VDCC是VDCC,VDCC是VDCC.芬太尼 (Fentanyl) 是一种药物.类阿片类受体 (MOR)疼痛 疼痛 疼痛 疼痛

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