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Updated: Jul 28, 2025

A Simple Bioassay for the Evaluation of Vascular Endothelial Growth Factors
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针对VEGFR-2的半合成抗癌神胺衍生物:在体和体外的评估

Mohammed A Dahab1, Hazem A Mahdy1, Hazem Elkady1

  • 1Pharmaceutical Medicinal Chemistry & Drug Design Department, Faculty of Pharmacy (Boys), Al-Azhar University, Cairo, Egypt.

Journal of biomolecular structure & dynamics
|June 1, 2023
PubMed
概括

新型神衍生物被设计为内皮生长因子受体-2 (VEGFR-2) 的抑制剂,用于治疗癌症. 化合物7g显示出强大的VEGFR-2抑制和显著的抗癌作用,显示出作为治疗剂的希望.

关键词:
这是一种抗癌药物.模拟MDMD的模拟在VEGFR-2的基础上,灭症 (apoptosis) 是一种死亡的过程.这是一种免疫调节剂.分子对接的分子对接.半合成是一种半合成.铁胺是什么意思 铁胺是什么意思

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