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Updated: Jul 28, 2025

Yeast Luminometric and Xenopus Oocyte Electrophysiological Examinations of the Molecular Mechanosensitivity of TRPV4
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暂时受体潜在氨酸1 (TRPA1) 调节剂:最近的更新和未来的前景

Zelin Hu1, Ya Zhang1, Wenhan Yu2

  • 1Department of Pulmonary and Critical Care Medicine, Targeted Tracer Research and Development Laboratory, Institute of Respiratory Health, Frontiers Science Center for Disease-related Molecular Network, National Clinical Research Center for Geriatrics, West China Hospital, Sichuan University, Chengdu, 610041, Sichuan, China; Precision Medicine Key Laboratory of Sichuan Province & Precision Medicine Research Center, West China Hospital, Sichuan University, Chengdu, 610041, Sichuan, China; College of Life Sciences, Sichuan University, Chengdu, 610064, China.

European journal of medicinal chemistry
|June 3, 2023
PubMed
概括

开发新的TRPA1调节器对于治疗疼痛,炎症和至关重要. 本综述侧重于最近的TRPA1抗剂和激动剂的结构-活性关系,以激发新的药物开发.

关键词:
激进主义者的激进主义者敌对者的敌对者离子通道 离子通道在 TRPA1 中,

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