Shohei Tsuchihashi1, Kazuma Nakashima1, Yuta Tarumizu2

  • 1Department of Patho-Functional Bioanalysis, Graduate School of Pharmaceutical Sciences, Kyoto University, 46-29 Yoshida Shimoadachi-cho, Sakyo-ku, Kyoto 606-8501, Japan.

概括

一种新的前列腺特异性膜抗原 (PSMA) 向剂,PSMA-NAT-DA1 (PNT-DA1),显示出增强的亲和力和瘤吸收. 这种PSMA放射性射剂在转移性割抵抗性前列腺癌的临床前模型中表现出优异的抗瘤作用.

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