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Updated: Jul 26, 2025

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埃拉克斯特兰的药理学和药理动力学

Jan H Beumer1,2,3, Julia Foldi4,5

  • 1Department of Pharmaceutical Sciences, School of Pharmacy, University of Pittsburgh, Pittsburgh, PA, 15261, USA. beumerj@gmail.com.

Cancer chemotherapy and pharmacology
|June 14, 2023
PubMed
概括

伊拉克斯特兰是一种口服选择性雌激素受体降解剂 (SERD),已获得FDA批准用于ER+/HER2-转移性乳腺癌与ESR1突变. 埃梅拉尔德试验显示了无进展生存率的改善,特别是在ESR1突变组.

关键词:
这种方法是Elacestrant.这就是Orserdu.药理动力学 药理动力学药理学 药理学 是一个学科.在RAD1901中,使用的是RAD1901.

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