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Updated: Jul 26, 2025

Microwave-Assisted Preparation of 1-Aryl-1H-pyrazole-5-amines
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合成,表征,抗结核活性和分子对接研究的Pyrazolylpyrazoline-Clubbed三醇和四醇混合物

Mayursinh Zala1, Jwalant J Vora1, Vijay M Khedkar2

  • 1Department of Chemistry, Faculty of Science, M.G. Science Institute, Affiliated with Gujarat University, Ahmedabad 380009, India.

ACS omega
|June 16, 2023
PubMed
概括

合成了新的pyrazolylpyrazoline衍生物,并对Mycobacterium tuberculosis进行了测试. 化合物9i,9k,9l,9o和9p显示出显著的抗结核活性,而化合物9o表现出最高的结合亲和力.

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