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Microwave-Assisted Preparation of 1-Aryl-1H-pyrazole-5-amines
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含有伊米达佐[2,1-b][1,3,4]蒂亚迪亚佐部分的皮拉衍生物的合成和抗菌活性评估

Jun-Da Qi1, Yu-Qing Meng2, Jingxin Sun1

  • 1Key Laboratory of Natural Medicines of the Changbai Mountain, Ministry of Education, College of Pharmacy, Yanbian University, Yanji, China.

Archiv der Pharmazie
|June 16, 2023
PubMed
概括

新型pyrazole衍生物显示出强大的抗真菌活性,其中化合物17l和17m显示出优越的疗效和低细胞毒性. 这些发现凸显了它们作为有前途的抗真菌剂的潜力.

关键词:
它是一种抗菌药物,具有抗菌作用.这是一种抗真菌药物.血液溶解 (hemolysis) 是一种皮拉 (pyrazole) 是一种可怕的药物.这种药物是提亚迪亚 (thiadiazole)

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