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大麻二醇通过两个不同的结合部位抑制Nav通道

Jian Huang1, Xiao Fan1, Xueqin Jin2

  • 1Department of Molecular Biology, Princeton University, Princeton, NJ, 08544, USA.

Nature communications
|June 17, 2023
PubMed
概括

大麻二醇 (CBD) 与通道Na1.7结合,稳定其无活化状态. 在特定结合部位的这一发现可能会导致新的疼痛和治疗方法.

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