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Updated: Jul 26, 2025

A High-Throughput Luciferase Assay to Evaluate Proteolysis of the Single-Turnover Protease PCSK9
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针对PCSK9来应对心血管疾病

Sandra Hummelgaard1, Joachim Pold Vilstrup2, Camilla Gustafsen2

  • 1Department of Biomedicine, Aarhus University, Aarhus, Denmark.

Pharmacology & therapeutics
|June 18, 2023
PubMed
概括

使用PCSK9抑制剂降低血胆固醇有效降低心血管疾病的风险. 这些疗法向PCSK9,这是LDL受体降解的关键调节者,为管理高胆固醇血症提供了一种新的方法.

关键词:
心血管疾病是什么心血管疾病降胆固醇剂可以降低胆固醇.这就是LDL-C.低密度脂蛋白受体的受体是低密度脂蛋白受体.在PCSK9中PCSK9 抑制剂的使用.

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