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对有机聚硫化物在人类TRPA1受体上的结合方式的阐释

Balázs Nemes1, Szabolcs László1,2, Balázs Zoltán Zsidó1

  • 1Department of Pharmacology and Pharmacotherapy, Medical School, University of Pécs, Pécs, Hungary.

Frontiers in physiology
|June 23, 2023
PubMed
概括

有机聚硫化物通过结合特定的氨酸残留物,主要是C621.1,激活TRPA1受体. 这一发现有助于开发用于缓解疼痛和炎症的新型TRPA1向药物.

关键词:
父亲们的父亲日期 时间 时间在DMTS中使用DMTS.绑定网站 绑定网站电友性TRPA1激动剂的电友性TRPA1激动剂.人类的TRPA1有机聚硫化物有机聚硫化物在位点导向的突变发生.

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