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Updated: Jul 25, 2025

A High-Throughput Luciferase Assay to Evaluate Proteolysis of the Single-Turnover Protease PCSK9
08:14

A High-Throughput Luciferase Assay to Evaluate Proteolysis of the Single-Turnover Protease PCSK9

Published on: August 28, 2018

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自然蛋白转化酶亚素/素9型抑制剂:一篇评论

Sonia Singh1, Himanshu Sharma2, Raghavan Ramankutty3

  • 1Institute of Pharmaceutical Research, GLA University, Mathura, U.P, 281406, India.

Combinatorial chemistry & high throughput screening
|June 27, 2023
PubMed
概括

目前正在探索天然存在的蛋白转化酶抑制剂亚素/素9型 (PCSK9) 抑制剂,以开发新的口服疗法. 这些化合物可以帮助更多的患者达到他们的LDL胆固醇目标,特别是当与他类药物一起使用时.

关键词:
紧急情况.急救.这就是为什么LDL,LDL是LDL.在PCSK9中胆固醇 胆固醇 胆固醇 是一种抑制剂 抑制剂 抑制剂一个单克隆抗体.

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