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Updated: Jul 25, 2025

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新型3,6-不和2,5-Diketopiperazines的设计,合成和抗癌活性

Xiaolin Li1,2, Tianrong Xun3, Huayan Xu4

  • 1Research Center for Marine Microbes, CAS Key Laboratory of Tropical Marine Bio-Resources and Ecology, Guangdong Key Laboratory of Marine Materia Medica, South China Sea Institute of Oceanology, Chinese Academy of Sciences, Guangzhou 510301, China.

Marine drugs
|June 27, 2023
PubMed
概括

新的二基托皮佩拉津衍生物被合成为潜在的抗癌剂. 化合物11对A549和Hela癌细胞表现出显著的活性,诱导细胞亡和阻断细胞循环的进展,表明其作为一种新的抗癌药物候选者的潜力.

关键词:
这是一种2,5-diketopiperazine衍生物.它具有抗癌活性,具有抗癌活性.电子的属性 电子的属性分子间的分子间键.脂溶性 脂溶性 脂溶性

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