新型α-Conotoxins的合成和生物活性来源于本土波利尼西亚形牛的新型α-Conotoxins

Yazid Mohamed Souf1, Gonxhe Lokaj2, Veeresh Kuruva3

  • 1CRIOBE, UAR CNRS-EPHE-UPVD 3278, Université de Perpignan Via Domitia, 58 Avenue Paul Alduy, 66860 Perpignan, France.

Marine drugs
|June 27, 2023
PubMed
概括

来自马奎萨斯群岛牛的两个新型α-conotoxins,GaIA和AdIA被合成和表征. 它们对大鼠尼古丁乙胆受体 (nAChRs) 具有强大的抑制活性,有助于理解nAChR亚型.

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