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Updated: Jul 24, 2025

Construction of Model Lipid Membranes Incorporating G-protein Coupled Receptors GPCRs
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在Gi-合受体GPR82处具有cationic头组的lysophospholipids的逆激素作用

Daisuke Yasuda1, Fumie Hamano2, Kazuyuki Masuda3

  • 1Department of Immunology, Graduate School of Medicine, Akita University, Akita, Japan.

European journal of pharmacology
|July 1, 2023
PubMed
概括

性溶解脂,包括埃德尔福辛,作为构成性活跃的GPR82受体的新型逆激动剂. 这些化合物抑制GPR82信号传递,并可能促进脂解.

关键词:
构成性活动 构成性活动在GPCR中,GPCR是指GPCR.反向激动剂是一种逆向激动剂.Lysophospholipid 是一种光脂的化合物.孤儿受体是一个孤儿受体.

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