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Updated: Jul 24, 2025

A Semi-High-Throughput Adaptation of the NADH-Coupled ATPase Assay for Screening Small Molecule Inhibitors
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针对actin N-终端乙转移酶NAA80的优化双基质抑制剂NAA80

Line M Myklebust1, Markus Baumann1,2, Svein I Støve1

  • 1Department of Biomedicine, University of Bergen, Bergen, Norway.

Frontiers in chemistry
|July 6, 2023
PubMed
概括

研究人员优化了一种新的NAA80酶抑制剂,CoA-Ac-EDDI-NH2,它针对actin的N终端乙化. 这种强大的化合物,IC50为120nM,有助于研究actin.

关键词:
在N端的乙化.NAA8080 NAA80808080 NAA808080 NAA808080 NAA80808080 NAA808080 NAA808080 NAA808080 NAA80808080 NAA808080 NAA808080 NAA808080 NAA808080 NAA8080 NAA8080 NAA8080 NAA8080 NAA8080 NAA8080 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80 NAA80乙烯基转移酶的使用方法这就是Actin Actin.这是一种双基质抑制剂.辅酶A 是一种细胞骨架 细胞骨架

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