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Updated: Jul 23, 2025

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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基于大麻素的类似物作为μ-阿片类受体的负基调节器的结构-活性关系研究

Taryn Bosquez-Berger1, Jessica A Gudorf2, Charles P Kuntz2

  • 1Gill Center for Biomolecular Science, Department of Psychological and Brain Sciences, Program in Neuroscience, Indiana University, Bloomington, Indiana 47405, United States.

Journal of medicinal chemistry
|July 12, 2023
PubMed
概括

基于大麻 (CBD) 的新药类相应物显示出对阿片类药物过量药物更强大的抗剂的希望. 这些化合物增强了纳洛对危险合成阿片类药物的有效性.

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