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Updated: Jul 23, 2025

Preparation of N-2-alkoxyvinylsulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines
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Preparation of N-2-alkoxyvinylsulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines

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二胺胺衍生物的二醇胺衍生物的碳酸胺酶抑制活性

Deepak Shilkar1, Mohd Usman Mohd Siddique2, Silvia Bua3

  • 1Department of Pharmaceutical Sciences and Technology, Birla Institute of Technology, Ranchi, India.

Journal of enzyme inhibition and medicinal chemistry
|July 13, 2023
PubMed
概括

甲胺覆盖的二胺被测试了碳酸无水酶的抑制. 化合物1显示出强烈的抑制人体碳酸无水酶I和II,表现优于乙胺.

关键词:
碳酸无水酶是一种碳酸无水酶.分子对接的分子对接.分子动力学分子动力学甲基硫甲基衍生物 甲基硫基衍生物

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