含有O-基-劳松与2-基基-β-环氧德克斯特林的复合物:制备,物理特征,抗寄生虫和抗真菌活性

Caroline Deckmann Nicoletti1, Raíssa Maria Dos Santos Galvão2, Marcella de Sá Haddad Queiroz1

  • 1Faculdade de Farmácia, Departamento de Tecnologia Farmacêutica, Universidade Federal Fluminense, 24241-000, Niterói, RJ, Brazil.

概括

将O-allyl-lawsone (OAL) 封装在2-hydroxypropyl-β-cyclodextrin (OAL MKN) 中可以增强其抗寄生虫和抗真菌活性. 这种OAL MKN配方显示出对Trypanosoma cruzi和Sporothrix酵母的有效性和选择性增加.

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