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Updated: Jul 19, 2025

Rapid In Situ Hybridization using Oligonucleotide Probes on Paraformaldehyde-prefixed Brain of Rats with Serotonin Syndrome
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2B确定:在药物发现中,色素受体2B的未来

Aaron M Bender1,2, Lauren C Parr1,2, William B Livingston3

  • 1Warren Center for Neuroscience Drug Discovery, Vanderbilt University, Nashville, Tennessee 37232, United States.

Journal of medicinal chemistry
|August 16, 2023
PubMed
概括

血清素5-HT2B受体激动剂引起心脏毒性,使其成为一个"抗目标". 然而,5-HT2B对抗剂在治疗肺动脉高血压和膜心脏病方面表现有前途.

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