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Updated: Jul 18, 2025

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作为COX抑制剂的新提亚碳胺衍生物:设计,合成,抗癌查,分子对接和ADME概况研究

Mohammed Hawash1, Nidal Jaradat1, Rozan Sabobeh1

  • 1Department of Pharmacy, Faculty of Medicine and Health Sciences, An-Najah National University, Nablus 400, Palestine.

ACS omega
|August 21, 2023
PubMed
概括

研究人员开发了新型的 thiazole carboxamide 衍生物来抑制循环氧化酶 (COX) 和抗癌. 化合物2b表现出强大的COX抑制和适度的抗癌作用,对正常细胞的毒性最小.

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