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Updated: Jul 18, 2025

Rapid Model to Evaluate the Anti-Obesity Potential of a Combination of Syzygium aromaticum Clove and Cuminun cyminum Cumin on C57BL6/j Mice Fed High-Fat Diet
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Rapid Model to Evaluate the Anti-Obesity Potential of a Combination of Syzygium aromaticum Clove and Cuminun cyminum Cumin on C57BL6/j Mice Fed High-Fat Diet

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大麻素类药物:设计比古安胺嵌入式,口服可用,外围选择性大麻素-1受体对手,用于代谢综合征障碍

Szabolcs Dvorácskó1,2, Alexa Herrerias3, Anna Oliverio3

  • 1Section on Medicinal Chemistry, National Institute on Alcohol Abuse and Alcoholism (NIAAA), National Institutes of Health (NIH), 5625 Fishers Lane, Rockville, Maryland 20852, United States.

Journal of medicinal chemistry
|August 23, 2023
PubMed
概括

开发了新的局限性大麻素-1受体 (CB1R) 抗剂. 这些化合物激活AMPK,在治疗肥胖和相关代谢障碍方面表现出有效性,对大脑的影响最小.

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