阻止CGRP受体:人类血管床之间的差异

Tessa de Vries1, Deirdre M Boucherie1, Antoon van den Bogaerdt2

  • 1Division of Vascular Medicine and Pharmacology, Department of Internal Medicine, Erasmus MC University Medical Center, P.O. Box 2040, 3000 CA Rotterdam, The Netherlands.

概括

扎维杰邦 (Zavegepant) 是一种小分子素基因相关 (CGRP) 受体对手,在人类冠状动脉和中脑膜动脉中表现出类似的效果. 这一发现对于评估新型偏头痛治疗的心血管安全性至关重要.

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