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Updated: Jul 16, 2025

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission

Published on: August 16, 2018

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发现和描述新型中枢神经系统透性GPR55抗原剂

Richard C Hewer1, Louisa A Christie1, Kevin J Doyle1

  • 1Cerevance Limited, 418 Cambridge Science Park, Cambridge CB4 0PZ, U.K.

Journal of medicinal chemistry
|September 14, 2023
PubMed
概括

研究人员确定G蛋白结合受体55 (GPR55) 是帕金森病运动症状的潜在目标. 开发了新的穿透大脑的GPR55激动剂,显示出选择性活性和进一步研究GPR55大脑功能的潜力.

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