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Updated: Jul 15, 2025

Author Spotlight: Investigating Physiological Functions of Vitamin A Transporters Using HPLC-Based Vitamin A Profiling
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开发酸受体α选择性对抗剂作为男性避孕药的新药的策略

Md Abdullah Al Noman1, Rebecca A D Cuellar1, Jillian L Kyzer1

  • 1Department of Medicinal Chemistry and Institute for Therapeutics Discovery and Development, College of Pharmacy, University of Minnesota, 717 Delaware Street SE, Minneapolis, MN, 55414, USA.

European journal of medicinal chemistry
|September 30, 2023
PubMed
概括

研究人员合成了26种视网氨酸类似物. 胺类同类型21显示出作为视网膜酸受体α对抗剂的潜力,但没有影响小鼠的雄性生育能力.

关键词:
男性的避孕药是男性的避孕药.网红酸受体α的受体是什么选择性的选择性结构与活动之间的关系.

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