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含有达沙替尼无水酸的口服配方改善了人类的可变性和生物可用性

Jiří Hofmann1, Aleš Bartůněk2, Tomáš Hauser1

  • 1Zentiva, k.s., Prague, Czech Republic.

Leukemia
|October 3, 2023
PubMed
概括

与慢性骨髓性白血病治疗的单酸形式相比,一种新的达沙替尼无水化合物配方显示出更好的吸收和降低的药物动力学变异性. 这一发展可能会导致更好的患者结果.

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