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Updated: Jul 14, 2025

Preparation of Enantiopure Non-Activated Aziridines and Synthesis of Biemamide B, D, and epiallo-Isomuscarine
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Preparation of Enantiopure Non-Activated Aziridines and Synthesis of Biemamide B, D, and epiallo-Isomuscarine

Published on: June 13, 2022

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合成和神经保护作用的3--3-乙烯基乙烯酸甲基衍生物的合成和神经保护作用

Urtė Šachlevičiūtė1, Gabriel Gonzalez2,3, Marie Kvasnicová2

  • 1Institute of Synthetic Chemistry, Kaunas University of Technology, Kaunas, Lithuania.

Archiv der Pharmazie
|October 5, 2023
PubMed
概括

研究人员开发了新型的阿兹提丁衍生物,具有治疗神经退行性疾病的巨大潜力. 几种化合物表现出类似于利瓦斯蒂格明的乙胆酶 (AChE) 抑制,其中28种化合物在帕金森病中表现出显著的神经保护作用.

关键词:
阿尔茨海默氏症是阿尔茨海默氏症的疾病帕金森病是帕金森病的一种疾病.乙烯基胆化酶的使用亚兹提丁胺是一种阿兹提丁胺.神经保护神经保护

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