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Updated: Jul 14, 2025

Pretargeted Radioimmunotherapy Based on the Inverse Electron Demand Diels-Alder Reaction
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抗瘤物质:过去,现在和未来?

Malcolm F G Stevens1, Richard T Wheelhouse2

  • 1Biodiscovery Institute, School of Pharmacy, University of Nottingham NG7 2RD UK.

RSC chemical biology
|October 6, 2023
PubMed
概括

40年来,人们已经知道像temozolomide这样的imidazotetrazines. 尽管它们在质瘤治疗中使用,但该化学类别的任何新药物都没有到达诊所.

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