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Updated: Jul 14, 2025

Reverse Yeast Two-hybrid System to Identify Mammalian Nuclear Receptor Residues that Interact with Ligands and/or Antagonists
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Piperlongumine 是孤儿核受体4A1 (NR4A1) 的一个配体

Lei Zhang1, Greg Martin1, Kumaravel Mohankumar1

  • 1Department of Veterinary Physiology and Pharmacology, Texas A&M University, College Station, TX, United States.

Frontiers in pharmacology
|October 9, 2023
PubMed
概括

作为一种抗癌药物,Piperlongumine通过诱导活性氧物种 (ROS) 和与NR4A1受体相互作用来抑制结肠癌细胞的生长. 这种机制为结肠癌治疗提供了一个新的治疗策略.

关键词:
没有4a1a1这就是ROSOS ROS.在TXNDC5中使用.癌症 癌症 癌症 癌症 癌症皮珀龙胺 (Piperlongumine) 是一种长胺.

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