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Updated: Jul 14, 2025

Achieving Efficient Fragment Screening at XChem Facility at Diamond Light Source
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Achieving Efficient Fragment Screening at XChem Facility at Diamond Light Source

Published on: May 29, 2021

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使用以功能为先的"侦察片段"为基础的方法,开发构造动态酶机械酶的全性共价抑制剂

Jared R Ramsey, Patrick M M Shelton, Tyler K Heiss

    bioRxiv : the preprint server for biology
    |October 9, 2023
    PubMed
    概括

    研究人员开发了一种新型的共价抑制剂策略,用于向酶,这是DNA/RNA重塑中的必不可少的酶. 这种方法利用了.

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