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来自Elephantopus scaber L.的结构多样化的类和它们的乙胆酶抑制活性

Jia-Yi Li1, Shu-Hui Dong1, Xin Zhang1

  • 1Key Laboratory of Computational Chemistry-Based Natural Antitumor Drug Research & Development, Liaoning Province; Engineering Research Center of Natural Medicine Active Molecule Research & Development, Liaoning Province; Key Laboratory of Natural Bioactive Compounds Discovery & Modification, Shenyang; School of Traditional Chinese Materia Medica, Shenyang Pharmaceutical University, Shenyang, Liaoning, 110016, China.

Phytochemistry
|October 9, 2023
PubMed
概括

从Elephantopus scaber L.中确定了三种新的化合物,即大象甲虫A-C. 大象虫B和C显示有前途的乙胆酶 (AChE) 抑制活性,表明潜在的治疗应用.

关键词:
乙胆化酶抑制剂 乙胆化酶抑制剂星座科 (Asteraceae) 是一个植物.埃莱芬托普斯 (Elephantopus scaber L. L.) 是一个大象食者.分子对接是分子对接.类物质是指类物质.

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