深入了解无处不在的脚手架Piperazine的结构-活动关系:一个解释性的审查

Jasmine Chaudhary1, Vishal Sharma1, Akash Jain1

  • 1Faculty of Pharmaceutical Sciences, M.M. College of Pharmacy, Maharishi Markandeshwer (Deemed to be University), Mullana, Ambala, Haryana, India.

概括

含有piperazine的药物具有广泛的治疗益处,但面临着耐受性和生物可用性差等挑战. 皮佩拉津支架的结构修改对于开发具有更高效率和亲和力的改进的候选药物至关重要.

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