化二甲基硫胺:分子建模,合成和试验室验证作为新的CETP抑制剂

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Reema Abu Khalaf1, Azhar Shalluf1, Maha Habash2

  • 1Department of Pharmacy, Faculty of Pharmacy, Al-Zaytoonah University of Jordan, Amman, Jordan.

Current computer-aided drug design
|October 19, 2023
PubMed
概括

新的二甲基硫胺被合成并测试了胆固醇转移蛋白 (CETP) 的抑制. 化合物7a-7g表现出强大的CETP抑制,为心血管疾病治疗提供了一个有前途的途径.

关键词:
胆固醇转移蛋白质的转移蛋白质迪亚利硫胺酸二甲酸超脂血症. 超脂血症. 这是一个很大的问题.利布多克 (Libdock) 是一种鱼类.连接 适合 适合制药剂的映射 制药剂的映射

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