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Updated: Jul 12, 2025

Solid-phase Synthesis of [4.4] Spirocyclic Oximes
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探索三环异环环作为RIOK2抑制剂的核心结构

Huilan Xiong1, Qiuchun Yu1, Haowen Ma1

  • 1International Cooperative Laboratory of Traditional Chinese Medicine Modernization and Innovative Drug Development, Ministry of Education (MOE) of People's Republic of China, College of Pharmacy, Jinan University 601 Huangpu Avenue West Guangzhou 510632 China weizhou088@jnu.edu.cn zhang_zhang@jnu.edu.cn caiqian@jnu.edu.cn.

RSC medicinal chemistry
|October 20, 2023
PubMed
概括

研究人员探索了RIOK2抑制剂的结构-活性关系. 合成了新的三环化合物,以了解CQ21111的结合重要性.

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