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Updated: Jul 12, 2025

Synthesis and Characterization of an Aspirin-fumarate Prodrug that Inhibits NFκB Activity and Breast Cancer Stem Cells
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作为抗癌和COX-2抑制剂的新型青混合物:合成,生物评估和对接研究

Mohammad Mahboob Alam1, Nawaf I Alsenani1, Antar A Abdelhamid1,2

  • 1Department of Chemistry, Faculty of Science, Al-Baha University, Al-Baha, Kingdom of Saudi Arabia.

Archiv der Pharmazie
|October 26, 2023
PubMed
概括

化学修饰的类醇衍生物显示出作为抗癌剂的前景. 化合物11有效地抑制了癌细胞生长和循环氧化酶-2 (COX-2) 活性,这表明了新的治疗途径.

关键词:
一,二,三三醇是什么一,三,四-氧化二醇.这是COX-2的代谢.这是一种抗癌药物.帕拉西托摩尔是一种可怕的药物.

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