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Updated: Jul 12, 2025

Microwave-Assisted Preparation of 1-Aryl-1H-pyrazole-5-amines
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新型抗结核剂:设计,合成,分子动力学和生物研究的Pyrazole - 1,2,4-Triazole结合物

K A Ajin1, Sethu Arun Kumar1, Manisha Singh1

  • 1Department of Pharmaceutical Chemistry, JSS College of Pharmacy, JSS Academy of Higher Education and Research, Sri Shivarathreeshwara Nagara, Mysuru, 570015, Karnataka, Indi.

Chemistry & biodiversity
|October 26, 2023
PubMed
概括

研究人员设计了针对DprE1酶的新型razol-linked triazoles,以对抗结核病. 几种化合物显示出显著的体外抗结核活性和低细胞毒性,表明可能成为新的抗结核药物.

关键词:
1,2,4-三醇是一种DprE1E1 的意思是什么?Mtb Mtb 在线观看这就是SBDDSBDD的意思.分子对接的分子对接.分子动态模拟分子动态模拟

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