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初级氨基的晚期同位素交换

Julia R Dorsheimer1, Tomislav Rovis1

  • 1Department of Chemistry, Columbia University, New York, New York 10027, United States.

Journal of the American Chemical Society
|October 27, 2023
PubMed
概括

研究人员开发了一种用于晚期同位素交换的新方法,使得-15 (15N) 标记的初级氨基的合成成为可能. 这一突破避免了药物发现中有价值的同位素的复杂新合成.

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