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Updated: Jul 12, 2025

Quantitative Structure-Activity Relationship, Activity Prediction, and Molecular Dynamics of Non-nucleotide Reverse Transcriptase Inhibitors
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Quantitative Structure-Activity Relationship, Activity Prediction, and Molecular Dynamics of Non-nucleotide Reverse Transcriptase Inhibitors

Published on: May 9, 2025

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设计和开发非核酸逆转录酶抑制剂 (NNRTIs) 的策略

Murugesan Vanangamudi1, Senthilkumar Palaniappan2,3, Muthu Kumaradoss Kathiravan4,5

  • 1Department of Pharmaceutical Chemistry, Amity Institute of Pharmacy, Amity University Madhya Pradesh, Gwalior 474005, Madhya Pradesh, India.

Viruses
|October 28, 2023
PubMed
概括

人类免疫缺陷病毒 (HIV) 导致艾滋病,这是全球卫生危机. 新的非核类逆转录酶抑制剂 (NNRTIs) 正在开发中,以对抗耐药性并提高艾滋病毒治疗疗效.

关键词:
艾滋病毒/艾滋病病毒/艾滋病病毒没有NNRTIs的NNRTI生物异构体替代药物卡特卡特是什么意思长效的注射剂 长效的注射剂分子混合化分子混合化.制药公司的药物战略.药物前体是药物前体.反向转录酶的使用在脚手架上跳跃跳跃.基于结构和片段的药物设计.

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